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Polycarboxylic fullerene derivatives as protein tyrosine phosphatase inhibitors

Oleksandr L Kobzar 1
Oleksandr L Kobzar
, 
Viacheslav V Trush 1
Viacheslav V Trush
, 
Vsevolod Yul'evich Tanchuk 1
Vsevolod Yul'evich Tanchuk
, 
Iliya Igorevich Voronov 2
Iliya Igorevich Voronov
, 
Aleksandr Sergeevich Peregudov 3
Aleksandr Sergeevich Peregudov
,  , 
Andriy I Vovk 1
Andriy I Vovk
10.1016/j.mencom.2015.05.013
Published 2015-04-28
Communication , Volume 25, Issue 3, 199-201
12
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Kobzar O. L. et al. Polycarboxylic fullerene derivatives as protein tyrosine phosphatase inhibitors // Mendeleev Communications. 2015. Vol. 25. No. 3. pp. 199-201.
GOST all authors (up to 50) Copy
Kobzar O. L., Trush V. V., Tanchuk V. Y., Voronov I. I., Peregudov A. S., Troshin P. A., Vovk A. I. Polycarboxylic fullerene derivatives as protein tyrosine phosphatase inhibitors // Mendeleev Communications. 2015. Vol. 25. No. 3. pp. 199-201.
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TY - JOUR
DO - 10.1016/j.mencom.2015.05.013
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2015.05.013
TI - Polycarboxylic fullerene derivatives as protein tyrosine phosphatase inhibitors
T2 - Mendeleev Communications
AU - Kobzar, Oleksandr L
AU - Trush, Viacheslav V
AU - Tanchuk, Vsevolod Yul'evich
AU - Voronov, Iliya Igorevich
AU - Peregudov, Aleksandr Sergeevich
AU - Troshin, Pavel Anatol'evich
AU - Vovk, Andriy I
PY - 2015
DA - 2015/04/28
PB - Mendeleev Communications
SP - 199-201
IS - 3
VL - 25
ER -
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@article{2015_Kobzar,
author = {Oleksandr L Kobzar and Viacheslav V Trush and Vsevolod Yul'evich Tanchuk and Iliya Igorevich Voronov and Aleksandr Sergeevich Peregudov and Pavel Anatol'evich Troshin and Andriy I Vovk},
title = {Polycarboxylic fullerene derivatives as protein tyrosine phosphatase inhibitors},
journal = {Mendeleev Communications},
year = {2015},
volume = {25},
publisher = {Mendeleev Communications},
month = {Apr},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2015.05.013},
number = {3},
pages = {199--201},
doi = {10.1016/j.mencom.2015.05.013}
}
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Kobzar, Oleksandr L., et al. “Polycarboxylic fullerene derivatives as protein tyrosine phosphatase inhibitors.” Mendeleev Communications, vol. 25, no. 3, Apr. 2015, pp. 199-201. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2015.05.013.

Abstract

The study of the inhibition of human protein tyrosine phosphatases by water-soluble [60]fullerene derivatives bearing five organic addends loaded with carboxylic groups demonstrated that a fullerene core is responsible for interactions with the enzymes while organic addends play a minor role modifying the selectivity of the inhibition.

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