Home / Publications / Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates

Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates

Rustam Rifkhatovich Davletshin
Marina Petrovna Shulaeva 2
Marina Petrovna Shulaeva
Kamil A. Ivshin 3
Kamil A. Ivshin
Natal'ya Victorovna Davletshina
Alexander Vladimirovich Gerasimov
Polina Aleksandrovna Kuryntseva
Sofia Vladimirovna Mosunova 1
Sofia Vladimirovna Mosunova
1 A. M. Butlerov Institute of Chemistry, Kazan Federal University, 420008 Kazan, Russian Federation
2 Kazan State Medical Academy, 420012 Kazan, Russian Federation
3 A. E. Arbuzov Institute of Organic and Physical Chemistry, FRC Kazan Scientific Center of the Russian Academy of Sciences, 420088 Kazan, Russian Federation
4 Institute of Biotechnology and Environmental Sciences, Kazan Federal University, 420088 Kazan, Russian Federation
Published 2025-02-18
CommunicationVolume 35, Issue 2, 152-154
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Davletshin R. R. et al. Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates // Mendeleev Communications. 2025. Vol. 35. No. 2. pp. 152-154.
GOST all authors (up to 50) Copy
Davletshin R. R., Sedov A. N., Shulaeva M. P., Ivshin K. A., Davletshina N. V., Gerasimov A. V., Kuryntseva P. A., Mosunova S. V. Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates // Mendeleev Communications. 2025. Vol. 35. No. 2. pp. 152-154.
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TY - JOUR
DO - 10.71267/mencom.7587
UR - https://mendcomm.colab.ws/publications/10.71267/mencom.7587
TI - Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates
T2 - Mendeleev Communications
AU - Davletshin, Rustam Rifkhatovich
AU - Sedov, Andrey Nikolaevich
AU - Shulaeva, Marina Petrovna
AU - Ivshin, Kamil A.
AU - Davletshina, Natal'ya Victorovna
AU - Gerasimov, Alexander Vladimirovich
AU - Kuryntseva, Polina Aleksandrovna
AU - Mosunova, Sofia Vladimirovna
PY - 2025
DA - 2025/02/18
PB - Mendeleev Communications
SP - 152-154
IS - 2
VL - 35
ER -
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@article{2025_Davletshin,
author = {Rustam Rifkhatovich Davletshin and Andrey Nikolaevich Sedov and Marina Petrovna Shulaeva and Kamil A. Ivshin and Natal'ya Victorovna Davletshina and Alexander Vladimirovich Gerasimov and Polina Aleksandrovna Kuryntseva and Sofia Vladimirovna Mosunova},
title = {Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates},
journal = {Mendeleev Communications},
year = {2025},
volume = {35},
publisher = {Mendeleev Communications},
month = {Feb},
url = {https://mendcomm.colab.ws/publications/10.71267/mencom.7587},
number = {2},
pages = {152--154},
doi = {10.71267/mencom.7587}
}
MLA
Cite this
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Davletshin, Rustam Rifkhatovich, et al. “Synthesis, structure and antimicrobial activity of dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates.” Mendeleev Communications, vol. 35, no. 2, Feb. 2025, pp. 152-154. https://mendcomm.colab.ws/publications/10.71267/mencom.7587.

Keywords

Abramov reaction
Antibacterial activity
Antifungal activity
solvent free conditions
X-ray diffraction.
α-hydroxy phosphonates

Abstract

New dialkyl [(hydroxy)(4-nitrophenyl)methyl]phosphonates containing various alkyl substituents were obtained from 4-nitrobenzaldehyde and the corresponding dialkyl phosphites and demonstrated antibacterial activity against Gram-positive bacterial strains B. cereus and S. aureus and antifungal activity against Candida albicans fungi. The dependence of antimicrobial activity on the nature of the substituents at the carbon atom a to phosphorus has been established.

Funders

Russian Science Foundation
24-23-00328

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