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Mild and regioselective straightforward synthesis of isomelatonin analogues

Eugene Pavlovich Zakurdaev 1
Eugene Pavlovich Zakurdaev
, 
Elizabeth Sergeevna Balenkova 1
Elizabeth Sergeevna Balenkova
, 
Valentin Georgievich Nenajdenko 1
Valentin Georgievich Nenajdenko
10.1070/MC2006v016n04ABEH002280
Published 2006-09-01
Communication , Volume 16, Issue 4, 213-215
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Zakurdaev E. P., Balenkova E. S., Nenajdenko V. G. Mild and regioselective straightforward synthesis of isomelatonin analogues // Mendeleev Communications. 2006. Vol. 16. No. 4. pp. 213-215.
GOST all authors (up to 50) Copy
Zakurdaev E. P., Balenkova E. S., Nenajdenko V. G. Mild and regioselective straightforward synthesis of isomelatonin analogues // Mendeleev Communications. 2006. Vol. 16. No. 4. pp. 213-215.
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TY - JOUR
DO - 10.1070/MC2006v016n04ABEH002280
UR - https://mendcomm.colab.ws/publications/10.1070/MC2006v016n04ABEH002280
TI - Mild and regioselective straightforward synthesis of isomelatonin analogues
T2 - Mendeleev Communications
AU - Zakurdaev, Eugene Pavlovich
AU - Balenkova, Elizabeth Sergeevna
AU - Nenajdenko, Valentin Georgievich
PY - 2006
DA - 2006/09/01
PB - Mendeleev Communications
SP - 213-215
IS - 4
VL - 16
ER -
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@article{2006_Zakurdaev,
author = {Eugene Pavlovich Zakurdaev and Elizabeth Sergeevna Balenkova and Valentin Georgievich Nenajdenko},
title = {Mild and regioselective straightforward synthesis of isomelatonin analogues},
journal = {Mendeleev Communications},
year = {2006},
volume = {16},
publisher = {Mendeleev Communications},
month = {Sep},
url = {https://mendcomm.colab.ws/publications/10.1070/MC2006v016n04ABEH002280},
number = {4},
pages = {213--215},
doi = {10.1070/MC2006v016n04ABEH002280}
}
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Zakurdaev, Eugene Pavlovich, et al. “Mild and regioselective straightforward synthesis of isomelatonin analogues.” Mendeleev Communications, vol. 16, no. 4, Sep. 2006, pp. 213-215. https://mendcomm.colab.ws/publications/10.1070/MC2006v016n04ABEH002280.

Abstract

A mild and regioselective strategy for 3-arylisomelatonins, compounds with prominent potential use as ligands for melatonin receptors, is developed.

References

1.
Do plasma melatonin concentrations decline with age?
Cornélissen G., Halberg F., Burioka N., Perfetto F., Tarquini R., Bakken E.E.
American Journal of Medicine, 2000
2.
Effects of melatonin on vascular reactivity, catecholamine levels, and blood pressure in healthy men.
Arangino S., Cagnacci A., Angiolucci M., Vacca A.M., Longu G., Volpe A., Melis G.B.
American Journal of Cardiology, 1999
3.
The Oxidant/Antioxidant Network: Role of Melatonin
Reiter R., Tan D., Cabrera J., D’Arpa D., Sainz R., Mayo J., Ramos S.
NeuroSignals, 1999
4.
Neuroprotective Effects of Melatonin
Lipartiti M., Franceschini D., Zanoni R., Gusella M., Giusti P., Cagnoli C.M., Kharlamov A., Manev H.
Advances in Experimental Medicine and Biology, 1996
5.
10.1070/MC2006v016n04ABEH002280_bib5_1
Blask
Cancer Res., 1997
8.
Melatonin Involvement in Immunity and Cancer
Fraschini F., Demartini G., Esposti D., Scaglione F.
NeuroSignals, 1998
9.
Synthesis and evaluation of a novel series of N,N-dimethylisotryptamines
Glennon R.A., Jacyno J.M., Young R., McKenney J.D., Nelson D.
Journal of Medicinal Chemistry, 1984
11.
2-Aryl tryptamines: selective high-affinity antagonists for the h5-HT2A receptor
Stevenson G.I., Smith A.L., Lewis S., Michie S.G., Neduvelil J.G., Patel S., Marwood R., Patel S., Castro J.L.
Bioorganic and Medicinal Chemistry Letters, 2000
12.
2-Substituted Tryptamines:  Agents with Selectivity for 5-HT6 Serotonin Receptors
Glennon R.A., Lee M., Rangisetty J.B., Dukat M., Roth B.L., Savage J.E., McBride A., Rauser L., Hufeisen S., Lee D.K.
Journal of Medicinal Chemistry, 2000
13.
Synthesis, pharmacological characterization and QSAR studies on 2-substituted indole melatonin receptor ligands
Mor M., Spadoni G., Di Giacomo B., Diamantini G., Bedini A., Tarzia G., Plazzi P.V., Rivara S., Nonno R., Lucini V., Pannacci M., Fraschini F., Stankov B.M.
Bioorganic and Medicinal Chemistry, 2001
14.
A convergent synthesis of (S)-β-methyl-2-aryltryptamine based gonadotropin releasing hormone antagonists
Walsh T.F., Toupence R.B., Ujjainwalla F., Young J.R., Goulet M.T.
Tetrahedron, 2001
15.
2-[N-Acylamino(C1−C3)alkyl]indoles as MT1 Melatonin Receptor Partial Agonists, Antagonists, and Putative Inverse Agonists
Spadoni G., Balsamini C., Bedini A., Diamantini G., Di Giacomo B., Tontini A., Tarzia G., Mor M., Plazzi P.V., Rivara S., Nonno R., Pannacci M., Lucini V., Fraschini F., Stankov B.M., et. al.
Journal of Medicinal Chemistry, 1998
16.
10.1070/MC2006v016n04ABEH002280_bib12
Shvedov
Khim. Geterotsikl. Soedin., 1973
17.
Convenient synthesis of melatonin analogues: 2- and 3-substituted -N-acetylindolylalkylamines
Nenajdenko V.G., Zakurdaev E.P., Prusov E.V., Balenkova E.S.
Tetrahedron, 2004
18.
The preparation of some thiochroman-3-ones and derivatives
Clark P.D., McKinnon D.M.
Canadian Journal of Chemistry, 1982
19.
Light-induced reactions of 2-(N-aikyi-N-arylamino)acetophenones and related amino-ketones: formation of 1,3-diarylazetidin-3-ols
Allworth K.L., El-Hamamy A.A., Hesabi M.M., Hill J.
Journal of the Chemical Society Perkin Transactions 1, 1980
20.
The preparation of some tetradecyl-substituted benzocarbazoles and benzacridines
Katritzky A.R., Wang Z., Savage G.P.
Journal of Heterocyclic Chemistry, 1991
22.
Indole aus cyclischen 1.3-Dicarbonylverbindungen mit substituierter 2-Stellung
Teuber H., Worbs E., Cornelius D.
Archiv der Pharmazie, 1982
23.
Structural problems in the indole group. Part V. Some derivatives of 2 : 3-diphenylindole
Coldham M.W., Lewis J.W., Plant S.G.
Journal of the Chemical Society (Resumed), 1954
24.
10.1070/MC2006v016n04ABEH002280_bib19
Grinev
Khim. -Pharm. Zh., 1984
25.
10.1070/MC2006v016n04ABEH002280_bib20
Bhattacharyya
Indian J. Chem., Sect. B., 1987
26.
Synthesis of 2,3-disubstituted indoles under mild conditions
Baccolini G., Todesco P.E.
Journal of the Chemical Society Chemical Communications, 1981
27.
Prochazka M.P., Eklund L., Carlson R., Hukkanen H., Nielsen M., Lehmann M.S., Tokii T.
Acta Chemica Scandinavica, 1990
28.
FISCHER INDOLE SYNTHESIS IN THE ABSENCE OF A SOLVENT
Matsumoto K., Tanaka A., Yukio I., Hayashi N., Toda M., Bulman R.A.
Heterocyclic Communications, 2003
29.
10.1070/MC2006v016n04ABEH002280_bib24
Letcher
J. Chem. Res., 1987
30.
621. Indoles. Part V. The Fischer cyclisation of some meta-substituted arylhydrazones
Ockenden D.W., Schofield K.
Journal of the Chemical Society (Resumed), 1957
31.
135. Dehydrogenation of tetrahydrocarbazoles by chloranil
Barclay B.M., Campbell N.
Journal of the Chemical Society (Resumed), 1945