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Synthesis of optically active imidazo[1,2-a]pyrimidin-3(2H)-ones

Mehdi Bakavoli 1
Mehdi Bakavoli
Ghodsieh Bagherzadeh 1
Ghodsieh Bagherzadeh
Mohammad Rahimizadeh 1
Mohammad Rahimizadeh
Published 2005-06-28
CommunicationVolume 15, Issue 4, 145-146
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Bakavoli M., Bagherzadeh G., Rahimizadeh M. Synthesis of optically active imidazo[1,2-a]pyrimidin-3(2H)-ones // Mendeleev Communications. 2005. Vol. 15. No. 4. pp. 145-146.
GOST all authors (up to 50) Copy
Bakavoli M., Bagherzadeh G., Rahimizadeh M. Synthesis of optically active imidazo[1,2-a]pyrimidin-3(2H)-ones // Mendeleev Communications. 2005. Vol. 15. No. 4. pp. 145-146.
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TY - JOUR
DO - 10.1070/MC2005v015n04ABEH001994
UR - https://mendcomm.colab.ws/publications/10.1070/MC2005v015n04ABEH001994
TI - Synthesis of optically active imidazo[1,2-a]pyrimidin-3(2H)-ones
T2 - Mendeleev Communications
AU - Bakavoli, Mehdi
AU - Bagherzadeh, Ghodsieh
AU - Rahimizadeh, Mohammad
PY - 2005
DA - 2005/06/28
PB - Mendeleev Communications
SP - 145-146
IS - 4
VL - 15
ER -
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@article{2005_Bakavoli,
author = {Mehdi Bakavoli and Ghodsieh Bagherzadeh and Mohammad Rahimizadeh},
title = {Synthesis of optically active imidazo[1,2-a]pyrimidin-3(2H)-ones},
journal = {Mendeleev Communications},
year = {2005},
volume = {15},
publisher = {Mendeleev Communications},
month = {Jun},
url = {https://mendcomm.colab.ws/publications/10.1070/MC2005v015n04ABEH001994},
number = {4},
pages = {145--146},
doi = {10.1070/MC2005v015n04ABEH001994}
}
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Bakavoli, Mehdi, et al. “Synthesis of optically active imidazo[1,2-a]pyrimidin-3(2H)-ones.” Mendeleev Communications, vol. 15, no. 4, Jun. 2005, pp. 145-146. https://mendcomm.colab.ws/publications/10.1070/MC2005v015n04ABEH001994.

Abstract

The reactions of 2-chloro-4-(substituted amino)-6-methyl-5-nitropyrimidine 1 with (L)-α-amino acids gave substituted derivatives 3, which were converted to optically active imidazo[1,2-a]pyrimidines 4 by treatment with either phosphorus oxychloride or polyphosphoric acid.

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