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Stable σ-adducts of 5-azauracil with C-nucleophiles

Yurii Alexeevich Azev 1
Yurii Alexeevich Azev
, 
Sergei Victorovich Shorshnev 2
Sergei Victorovich Shorshnev
, 
Detlef Gabel 3
Detlef Gabel
1 Ural Scientific Research Institute of Technology of Medical Preparations, Ekaterinburg, Russian Federation
2 ChemBridge, Moscow, Russian Federation
10.1070/MC2001v011n06ABEH001508
Published 2001-12-18
Communication , Volume 11, Issue 6, 234-235
5
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Azev Y. A., Shorshnev S. V., Gabel D. Stable σ-adducts of 5-azauracil with C-nucleophiles // Mendeleev Communications. 2001. Vol. 11. No. 6. pp. 234-235.
GOST all authors (up to 50) Copy
Azev Y. A., Shorshnev S. V., Gabel D. Stable σ-adducts of 5-azauracil with C-nucleophiles // Mendeleev Communications. 2001. Vol. 11. No. 6. pp. 234-235.
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TY - JOUR
DO - 10.1070/MC2001v011n06ABEH001508
UR - https://mendcomm.colab.ws/publications/10.1070/MC2001v011n06ABEH001508
TI - Stable σ-adducts of 5-azauracil with C-nucleophiles
T2 - Mendeleev Communications
AU - Azev, Yurii Alexeevich
AU - Shorshnev, Sergei Victorovich
AU - Gabel, Detlef
PY - 2001
DA - 2001/12/18
PB - Mendeleev Communications
SP - 234-235
IS - 6
VL - 11
ER -
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@article{2001_Azev,
author = {Yurii Alexeevich Azev and Sergei Victorovich Shorshnev and Detlef Gabel},
title = {Stable σ-adducts of 5-azauracil with C-nucleophiles},
journal = {Mendeleev Communications},
year = {2001},
volume = {11},
publisher = {Mendeleev Communications},
month = {Dec},
url = {https://mendcomm.colab.ws/publications/10.1070/MC2001v011n06ABEH001508},
number = {6},
pages = {234--235},
doi = {10.1070/MC2001v011n06ABEH001508}
}
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Azev, Yurii Alexeevich, et al. “Stable σ-adducts of 5-azauracil with C-nucleophiles.” Mendeleev Communications, vol. 11, no. 6, Dec. 2001, pp. 234-235. https://mendcomm.colab.ws/publications/10.1070/MC2001v011n06ABEH001508.

Abstract

The heating of 5-azauracil 1 with malonamide in butanol resulted in 1,2,3,4,5,6-hexahydro-6-(dicarbamoylmethyl)-1,3,5-triazine- 2,4-dione 3. Under conditions of acid catalysis, compound 1 reacted with o-phenylenediamine, pyrrogallol, resorcinol and phenylhydrazine derivatives to form the corresponding 6-derivatives of 1,2,3,4,5,6-hexahydro-1,3,5-triazine-2,4-dione.

References

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Chung W.K., Chung J.H., Watanabe K.A.
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10.1070/MC2001v011n06ABEH001508_bib4
van der Plas
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