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New approach to [a]-fused fluoroquinolones: the synthesis of 5-oxo-1,2,3,3a,4,5-hexahydropyrrolo[1,2-a]quinolines

Elizaveta Vladimirovna Tsoi 1
Elizaveta Vladimirovna Tsoi
,  , 
Emiliya Vladimirovna Nosova 1
Emiliya Vladimirovna Nosova
, 
Galina Nikolaevna Lipunova 1
Galina Nikolaevna Lipunova
, 
Alexey Vasil'evich Tkachev 2
Alexey Vasil'evich Tkachev
10.1070/MC2001v011n02ABEH001323
Published 2001-04-24
Communication , Volume 11, Issue 2, 53-54
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Tsoi E. V. et al. New approach to [a]-fused fluoroquinolones: the synthesis of 5-oxo-1,2,3,3a,4,5-hexahydropyrrolo[1,2-a]quinolines // Mendeleev Communications. 2001. Vol. 11. No. 2. pp. 53-54.
GOST all authors (up to 50) Copy
Tsoi E. V., Charushin V. N., Nosova E. V., Lipunova G. N., Tkachev A. V. New approach to [a]-fused fluoroquinolones: the synthesis of 5-oxo-1,2,3,3a,4,5-hexahydropyrrolo[1,2-a]quinolines // Mendeleev Communications. 2001. Vol. 11. No. 2. pp. 53-54.
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TY - JOUR
DO - 10.1070/MC2001v011n02ABEH001323
UR - https://mendcomm.colab.ws/publications/10.1070/MC2001v011n02ABEH001323
TI - New approach to [a]-fused fluoroquinolones: the synthesis of 5-oxo-1,2,3,3a,4,5-hexahydropyrrolo[1,2-a]quinolines
T2 - Mendeleev Communications
AU - Tsoi, Elizaveta Vladimirovna
AU - Charushin, Valery Nikolaevich
AU - Nosova, Emiliya Vladimirovna
AU - Lipunova, Galina Nikolaevna
AU - Tkachev, Alexey Vasil'evich
PY - 2001
DA - 2001/04/24
PB - Mendeleev Communications
SP - 53-54
IS - 2
VL - 11
ER -
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@article{2001_Tsoi,
author = {Elizaveta Vladimirovna Tsoi and Valery Nikolaevich Charushin and Emiliya Vladimirovna Nosova and Galina Nikolaevna Lipunova and Alexey Vasil'evich Tkachev},
title = {New approach to [a]-fused fluoroquinolones: the synthesis of 5-oxo-1,2,3,3a,4,5-hexahydropyrrolo[1,2-a]quinolines},
journal = {Mendeleev Communications},
year = {2001},
volume = {11},
publisher = {Mendeleev Communications},
month = {Apr},
url = {https://mendcomm.colab.ws/publications/10.1070/MC2001v011n02ABEH001323},
number = {2},
pages = {53--54},
doi = {10.1070/MC2001v011n02ABEH001323}
}
MLA
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Tsoi, Elizaveta Vladimirovna, et al. “New approach to [a]-fused fluoroquinolones: the synthesis of 5-oxo-1,2,3,3a,4,5-hexahydropyrrolo[1,2-a]quinolines.” Mendeleev Communications, vol. 11, no. 2, Apr. 2001, pp. 53-54. https://mendcomm.colab.ws/publications/10.1070/MC2001v011n02ABEH001323.

Abstract

The reaction of N-(ethoxycarbonyl)methyl substituted ethyl 6,7-difluoro-, 6,7,8-trifluoro- and 5,6,7,8-tetrafluoro-4-oxo-1,4-dihydroquinoline-3-carboxylates with methyl methacrylate results in the [3 + 2] adducts, hexahydropyrrolo[1,2-a]quinolones, which can be precursors of [a]-fused fluoroquinolones.

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