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Synthesis of hybrid molecules based on thioglycolurils and 1,2,5-oxadiazoles via the Eschenmoser sulfide contraction

Ekaterina Evgenievna Vinogradova 1
Ekaterina Evgenievna Vinogradova
Alexander Aleksandrovich Larin
Galina Anatol'evna Gazieva 1
Galina Anatol'evna Gazieva
Published 2023-12-25
CommunicationVolume 34, Issue 1, 122-125
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Vinogradova E. E., Larin A. A., Gazieva G. A. Synthesis of hybrid molecules based on thioglycolurils and 1,2,5-oxadiazoles via the Eschenmoser sulfide contraction // Mendeleev Communications. 2023. Vol. 34. No. 1. pp. 122-125.
GOST all authors (up to 50) Copy
Vinogradova E. E., Larin A. A., Gazieva G. A. Synthesis of hybrid molecules based on thioglycolurils and 1,2,5-oxadiazoles via the Eschenmoser sulfide contraction // Mendeleev Communications. 2023. Vol. 34. No. 1. pp. 122-125.
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TY - JOUR
DO - 10.1016/j.mencom.2024.01.037
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2024.01.037
TI - Synthesis of hybrid molecules based on thioglycolurils and 1,2,5-oxadiazoles via the Eschenmoser sulfide contraction
T2 - Mendeleev Communications
AU - Vinogradova, Ekaterina Evgenievna
AU - Larin, Alexander Aleksandrovich
AU - Gazieva, Galina Anatol'evna
PY - 2023
DA - 2023/12/25
PB - Mendeleev Communications
SP - 122-125
IS - 1
VL - 34
ER -
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@article{2023_Vinogradova,
author = {Ekaterina Evgenievna Vinogradova and Alexander Aleksandrovich Larin and Galina Anatol'evna Gazieva},
title = {Synthesis of hybrid molecules based on thioglycolurils and 1,2,5-oxadiazoles via the Eschenmoser sulfide contraction},
journal = {Mendeleev Communications},
year = {2023},
volume = {34},
publisher = {Mendeleev Communications},
month = {Dec},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2024.01.037},
number = {1},
pages = {122--125},
doi = {10.1016/j.mencom.2024.01.037}
}
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Vinogradova, Ekaterina Evgenievna, et al. “Synthesis of hybrid molecules based on thioglycolurils and 1,2,5-oxadiazoles via the Eschenmoser sulfide contraction.” Mendeleev Communications, vol. 34, no. 1, Dec. 2023, pp. 122-125. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2024.01.037.
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Keywords

Eschenmoser sulfide contraction.
furazan
furoxan
glycoluril
thioglycoluril

Abstract

A simple synthesis of novel hybrid molecules containing methylidenehexahydroimidazo[4,5-d]imidazol-2(1H)-one and 1,2,5-oxadiazole moieties is based on the Eschenmoser sulfide contraction involving alkylative precoupling of thioglycolurils with 3(4)-bromoacetyl-1,2,5-oxadiazoles. The proposed method does not require using toxic PPh3 for sulfur extrusion. The synthesized compounds may serve as platforms for constructing both new bioactive and new high- energy compounds.

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