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Novel sulfamoylbenzoates as antifungal agents against Malassezia furfur

Lena Trifonov 1
Lena Trifonov
, 
Katerina Chumin 2
Katerina Chumin
, 
Raanan Gvirtz 1, 2
Raanan Gvirtz
, 
Michal Afri 1
Michal Afri
, 
Edward E Korshin 1
Edward E Korshin
, 
Guy Cohen 2
Guy Cohen
, 
Arie Gruzman 1
Arie Gruzman
2 The Skin Research Institute, The Dead-Sea and Arava Science Center, Masada, Israel
10.1016/j.mencom.2020.11.006
Published 2020-11-03
Communication , Volume 30, Issue 6, 709-711
2
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Trifonov L. et al. Novel sulfamoylbenzoates as antifungal agents against Malassezia furfur // Mendeleev Communications. 2020. Vol. 30. No. 6. pp. 709-711.
GOST all authors (up to 50) Copy
Trifonov L., Chumin K., Gvirtz R., Afri M., Korshin E. E., Cohen G., Gruzman A. Novel sulfamoylbenzoates as antifungal agents against Malassezia furfur // Mendeleev Communications. 2020. Vol. 30. No. 6. pp. 709-711.
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TY - JOUR
DO - 10.1016/j.mencom.2020.11.006
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2020.11.006
TI - Novel sulfamoylbenzoates as antifungal agents against Malassezia furfur
T2 - Mendeleev Communications
AU - Trifonov, Lena
AU - Chumin, Katerina
AU - Gvirtz, Raanan
AU - Afri, Michal
AU - Korshin, Edward E
AU - Cohen, Guy
AU - Gruzman, Arie
PY - 2020
DA - 2020/11/03
PB - Mendeleev Communications
SP - 709-711
IS - 6
VL - 30
ER -
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@article{2020_Trifonov,
author = {Lena Trifonov and Katerina Chumin and Raanan Gvirtz and Michal Afri and Edward E Korshin and Guy Cohen and Arie Gruzman},
title = {Novel sulfamoylbenzoates as antifungal agents against Malassezia furfur},
journal = {Mendeleev Communications},
year = {2020},
volume = {30},
publisher = {Mendeleev Communications},
month = {Nov},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2020.11.006},
number = {6},
pages = {709--711},
doi = {10.1016/j.mencom.2020.11.006}
}
MLA
Cite this
MLA Copy
Trifonov, Lena, et al. “Novel sulfamoylbenzoates as antifungal agents against Malassezia furfur.” Mendeleev Communications, vol. 30, no. 6, Nov. 2020, pp. 709-711. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2020.11.006.

Keywords

Malassezia furfur
arenesulfonamides
fungicides
medicinal chemistry
seborrheic dermatitis

Abstract

Novel polyfunctional arenesulfonamides as potential fungicides were prepared in eight steps from 3-amino-5-bromobenzoic acid. Among them, methyl 3-bromo-2-nitro-5-(N-phenylsulfamoyl)benzoate exhibiting significant cytotoxic activity against Malassezia furfur is proposed as a lead for the development of drug candidates against skin diseases caused by the fungi, especially against seborrheic dermatitis.

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