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Synthesis and biological evaluation of novel bispyridinium salts containing naphthalene-2,7-diylbis(oxy) spacer

Anatoly Nikolaevich Vereshchagin 1
Anatoly Nikolaevich Vereshchagin
, 
Nikita Andreevich Frolov 1
Nikita Andreevich Frolov
, 
Anna S Pakina 1, 2
Anna S Pakina
, 
Karl A Hansford 3
Karl A Hansford
, 
Mikhail Petrovich Egorov 1
Mikhail Petrovich Egorov
10.1016/j.mencom.2020.11.004
Published 2020-11-03
Communication , Volume 30, Issue 6, 703-705
9
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Vereshchagin A. N. et al. Synthesis and biological evaluation of novel bispyridinium salts containing naphthalene-2,7-diylbis(oxy) spacer // Mendeleev Communications. 2020. Vol. 30. No. 6. pp. 703-705.
GOST all authors (up to 50) Copy
Vereshchagin A. N., Frolov N. A., Pakina A. S., Hansford K. A., Egorov M. P. Synthesis and biological evaluation of novel bispyridinium salts containing naphthalene-2,7-diylbis(oxy) spacer // Mendeleev Communications. 2020. Vol. 30. No. 6. pp. 703-705.
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TY - JOUR
DO - 10.1016/j.mencom.2020.11.004
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2020.11.004
TI - Synthesis and biological evaluation of novel bispyridinium salts containing naphthalene-2,7-diylbis(oxy) spacer
T2 - Mendeleev Communications
AU - Vereshchagin, Anatoly Nikolaevich
AU - Frolov, Nikita Andreevich
AU - Pakina, Anna S
AU - Hansford, Karl A
AU - Egorov, Mikhail Petrovich
PY - 2020
DA - 2020/11/03
PB - Mendeleev Communications
SP - 703-705
IS - 6
VL - 30
ER -
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@article{2020_Vereshchagin,
author = {Anatoly Nikolaevich Vereshchagin and Nikita Andreevich Frolov and Anna S Pakina and Karl A Hansford and Mikhail Petrovich Egorov},
title = {Synthesis and biological evaluation of novel bispyridinium salts containing naphthalene-2,7-diylbis(oxy) spacer},
journal = {Mendeleev Communications},
year = {2020},
volume = {30},
publisher = {Mendeleev Communications},
month = {Nov},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2020.11.004},
number = {6},
pages = {703--705},
doi = {10.1016/j.mencom.2020.11.004}
}
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Vereshchagin, Anatoly Nikolaevich, et al. “Synthesis and biological evaluation of novel bispyridinium salts containing naphthalene-2,7-diylbis(oxy) spacer.” Mendeleev Communications, vol. 30, no. 6, Nov. 2020, pp. 703-705. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2020.11.004.

Keywords

antibacterial agents
Antifungal activity
biological activity
bis-quaternary ammonium compounds
pyridinium salts

Abstract

Novel five bispyridinium salts based on a naphthalene-2,7-diylbis(oxy) spacer were synthesized. The obtained compounds showed stronger biological activity against five strains of bacteria and two fungi as compared to modern biocides used in the pharmaceutical market.

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