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Synthesis of potential anti-Trypanosoma cruzi azole-naftifine analogues by azide–alkyne click reaction

Carlos Henrique Callegario Zacchi 1
Carlos Henrique Callegario Zacchi
, 
Stephanie Souto Maior Federighi 2
Stephanie Souto Maior Federighi
, 
Fernanda Ramos Gadelha 2
Fernanda Ramos Gadelha
, 
Felipe Terra Martins 3
Felipe Terra Martins
, 
Rosemeire Brondi Alves 1
Rosemeire Brondi Alves
, 
Ângelo de Fátima 1
Ângelo de Fátima
10.1016/j.mencom.2018.03.029
Published 2018-03-01
Communication , Volume 28, Issue 2, 195-197
3
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Zacchi C. H. C. et al. Synthesis of potential anti-Trypanosoma cruzi azole-naftifine analogues by azide–alkyne click reaction // Mendeleev Communications. 2018. Vol. 28. No. 2. pp. 195-197.
GOST all authors (up to 50) Copy
Zacchi C. H. C., Federighi S. S. M., Gadelha F. R., Martins F. T., Alves R. B., de Fátima Â. Synthesis of potential anti-Trypanosoma cruzi azole-naftifine analogues by azide–alkyne click reaction // Mendeleev Communications. 2018. Vol. 28. No. 2. pp. 195-197.
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TY - JOUR
DO - 10.1016/j.mencom.2018.03.029
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2018.03.029
TI - Synthesis of potential anti-Trypanosoma cruzi azole-naftifine analogues by azide–alkyne click reaction
T2 - Mendeleev Communications
AU - Zacchi, Carlos Henrique Callegario
AU - Federighi, Stephanie Souto Maior
AU - Gadelha, Fernanda Ramos
AU - Martins, Felipe Terra
AU - Alves, Rosemeire Brondi
AU - de Fátima, Ângelo
PY - 2018
DA - 2018/03/01
PB - Mendeleev Communications
SP - 195-197
IS - 2
VL - 28
ER -
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@article{2018_Zacchi,
author = {Carlos Henrique Callegario Zacchi and Stephanie Souto Maior Federighi and Fernanda Ramos Gadelha and Felipe Terra Martins and Rosemeire Brondi Alves and Ângelo de Fátima},
title = {Synthesis of potential anti-Trypanosoma cruzi azole-naftifine analogues by azide–alkyne click reaction},
journal = {Mendeleev Communications},
year = {2018},
volume = {28},
publisher = {Mendeleev Communications},
month = {Mar},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2018.03.029},
number = {2},
pages = {195--197},
doi = {10.1016/j.mencom.2018.03.029}
}
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Zacchi, Carlos Henrique Callegario, et al. “Synthesis of potential anti-Trypanosoma cruzi azole-naftifine analogues by azide–alkyne click reaction.” Mendeleev Communications, vol. 28, no. 2, Mar. 2018, pp. 195-197. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2018.03.029.

Abstract

Twenty novel azole-naftifine analogues were obtained using azide–alkyne click reaction. Five of them were more potent than the positive control naftifine revealing an unprecedented antiproliferative effects against Trypanosoma cruzi.

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