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β-d-Ribofuranosyl substituted polyfluoroalkylpyrazoles and their activity against the influenza virus

Anna Evgen'evna Ivanova 1
Anna Evgen'evna Ivanova
, 
Yanina Valer'evna Burgart 1
Yanina Valer'evna Burgart
, 
Viktor Ivanovich Saloutin 1
Viktor Ivanovich Saloutin
, 
Yana R Orshanskaya 2
Yana R Orshanskaya
, 
Vladimir Victorovich Zarubaev 2
Vladimir Victorovich Zarubaev
10.1016/j.mencom.2018.01.017
Published 2017-12-22
Communication , Volume 28, Issue 1, 52-54
9
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Ivanova A. E. et al. β-d-Ribofuranosyl substituted polyfluoroalkylpyrazoles and their activity against the influenza virus // Mendeleev Communications. 2017. Vol. 28. No. 1. pp. 52-54.
GOST all authors (up to 50) Copy
Ivanova A. E., Burgart Y. V., Saloutin V. I., Orshanskaya Y. R., Zarubaev V. V. β-d-Ribofuranosyl substituted polyfluoroalkylpyrazoles and their activity against the influenza virus // Mendeleev Communications. 2017. Vol. 28. No. 1. pp. 52-54.
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TY - JOUR
DO - 10.1016/j.mencom.2018.01.017
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2018.01.017
TI - β-d-Ribofuranosyl substituted polyfluoroalkylpyrazoles and their activity against the influenza virus
T2 - Mendeleev Communications
AU - Ivanova, Anna Evgen'evna
AU - Burgart, Yanina Valer'evna
AU - Saloutin, Viktor Ivanovich
AU - Orshanskaya, Yana R
AU - Zarubaev, Vladimir Victorovich
PY - 2017
DA - 2017/12/22
PB - Mendeleev Communications
SP - 52-54
IS - 1
VL - 28
ER -
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@article{2017_Ivanova,
author = {Anna Evgen'evna Ivanova and Yanina Valer'evna Burgart and Viktor Ivanovich Saloutin and Yana R Orshanskaya and Vladimir Victorovich Zarubaev},
title = {β-d-Ribofuranosyl substituted polyfluoroalkylpyrazoles and their activity against the influenza virus},
journal = {Mendeleev Communications},
year = {2017},
volume = {28},
publisher = {Mendeleev Communications},
month = {Dec},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2018.01.017},
number = {1},
pages = {52--54},
doi = {10.1016/j.mencom.2018.01.017}
}
MLA
Cite this
MLA Copy
Ivanova, Anna Evgen'evna, et al. “β-d-Ribofuranosyl substituted polyfluoroalkylpyrazoles and their activity against the influenza virus.” Mendeleev Communications, vol. 28, no. 1, Dec. 2017, pp. 52-54. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2018.01.017.

Abstract

Regiospecific ribosylation of 3-polyfluoroalkyl-5-phenylpyrazoles with 1,2,3,5-tetra-O-acetyl-β-d-ribofuranose in the presence of tin(iv) chloride followed by deacetylation affords 1-(β-d-ribofuranosyl)-3-polyfluoroalkyl-5-phenyl- 1H-pyrazoles. These derivatives as well as starting pyrazoles were tested for anti-influenza activity.

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