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New benzophenone phosphonate derivatives

Maxim Sergeevich Gaman 1
Maxim Sergeevich Gaman
, 
Elena Sergeevna Matyugina 1
Elena Sergeevna Matyugina
, 
Mikhail Stanislavovich Novikov 2
Mikhail Stanislavovich Novikov
, 
Denis Aleksandrovich Babkov 2
Denis Aleksandrovich Babkov
,  , 
Sergei Nikolaevich Kochetkov 1
Sergei Nikolaevich Kochetkov
, 
Anastasia Lvovna Khandazhinskaya 1
Anastasia Lvovna Khandazhinskaya
10.1016/j.mencom.2017.07.008
Published 2017-06-29
Communication , Volume 27, Issue 4, 346-348
2
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Gaman M. S. et al. New benzophenone phosphonate derivatives // Mendeleev Communications. 2017. Vol. 27. No. 4. pp. 346-348.
GOST all authors (up to 50) Copy
Gaman M. S., Matyugina E. S., Novikov M. S., Babkov D. A., Solyev P. N., Kochetkov S. N., Khandazhinskaya A. L. New benzophenone phosphonate derivatives // Mendeleev Communications. 2017. Vol. 27. No. 4. pp. 346-348.
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TY - JOUR
DO - 10.1016/j.mencom.2017.07.008
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2017.07.008
TI - New benzophenone phosphonate derivatives
T2 - Mendeleev Communications
AU - Gaman, Maxim Sergeevich
AU - Matyugina, Elena Sergeevna
AU - Novikov, Mikhail Stanislavovich
AU - Babkov, Denis Aleksandrovich
AU - Solyev, Pavel Nikolayevich
AU - Kochetkov, Sergei Nikolaevich
AU - Khandazhinskaya, Anastasia Lvovna
PY - 2017
DA - 2017/06/29
PB - Mendeleev Communications
SP - 346-348
IS - 4
VL - 27
ER -
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@article{2017_Gaman,
author = {Maxim Sergeevich Gaman and Elena Sergeevna Matyugina and Mikhail Stanislavovich Novikov and Denis Aleksandrovich Babkov and Pavel Nikolayevich Solyev and Sergei Nikolaevich Kochetkov and Anastasia Lvovna Khandazhinskaya},
title = {New benzophenone phosphonate derivatives},
journal = {Mendeleev Communications},
year = {2017},
volume = {27},
publisher = {Mendeleev Communications},
month = {Jun},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2017.07.008},
number = {4},
pages = {346--348},
doi = {10.1016/j.mencom.2017.07.008}
}
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Gaman, Maxim Sergeevich, et al. “New benzophenone phosphonate derivatives.” Mendeleev Communications, vol. 27, no. 4, Jun. 2017, pp. 346-348. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2017.07.008.

Abstract

New well-soluble in 10% DMSO phosphonate derivatives of substituted benzophenone have been synthesized using different methods. Preliminary computer modeling of proposed structures in the reverse transcriptase HIV-1 hydrophobic pocket suggested these molecules as potential non-nucleoside inhibitors of this enzyme.

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Vogel's Textbook of Practical Organic Chemistry, 1989