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One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids

Sergei Valentinovich Baikov 1
Sergei Valentinovich Baikov
, 
Galina Grigor'evna Krasovskaya 1
Galina Grigor'evna Krasovskaya
, 
Alexei Vladislavovich Kolobov 1
Alexei Vladislavovich Kolobov
, 
Evgenii Romanovich Kofanov 1
Evgenii Romanovich Kofanov
10.1016/j.mencom.2015.03.021
Published 2015-03-06
Communication , Volume 25, Issue 2, 138-139
2
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Baikov S. V. et al. One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids // Mendeleev Communications. 2015. Vol. 25. No. 2. pp. 138-139.
GOST all authors (up to 50) Copy
Baikov S. V., Krasovskaya G. G., Kolobov A. V., Kofanov E. R. One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids // Mendeleev Communications. 2015. Vol. 25. No. 2. pp. 138-139.
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TY - JOUR
DO - 10.1016/j.mencom.2015.03.021
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2015.03.021
TI - One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids
T2 - Mendeleev Communications
AU - Baikov, Sergei Valentinovich
AU - Krasovskaya, Galina Grigor'evna
AU - Kolobov, Alexei Vladislavovich
AU - Kofanov, Evgenii Romanovich
PY - 2015
DA - 2015/03/06
PB - Mendeleev Communications
SP - 138-139
IS - 2
VL - 25
ER -
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@article{2015_Baikov,
author = {Sergei Valentinovich Baikov and Galina Grigor'evna Krasovskaya and Alexei Vladislavovich Kolobov and Evgenii Romanovich Kofanov},
title = {One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids},
journal = {Mendeleev Communications},
year = {2015},
volume = {25},
publisher = {Mendeleev Communications},
month = {Mar},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2015.03.021},
number = {2},
pages = {138--139},
doi = {10.1016/j.mencom.2015.03.021}
}
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Baikov, Sergei Valentinovich, et al. “One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids.” Mendeleev Communications, vol. 25, no. 2, Mar. 2015, pp. 138-139. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2015.03.021.

Abstract

Heterocyclization of toluic acid amidoximes with acetic or propionic anhydrides affords 5-alkyl-3-tolyl-1,2,4-oxadiazoles, whose air oxidation in the same vessel gives (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids.

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