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Novel synthetic routes to N-(2-amino-9H-purin-6-yl)-substituted amino acids

Alexey Yur'evich Vigorov 1
Alexey Yur'evich Vigorov
, 
Victor Pavlovich Krasnov 1
Victor Pavlovich Krasnov
, 
Dmitry Andreevich Gruzdev 1
Dmitry Andreevich Gruzdev
, 
Alisa A Men'shikova 1
Alisa A Men'shikova
, 
Alexander Mikhailovich Demin 1
Alexander Mikhailovich Demin
, 
Galina L'vovna Levit 1
Galina L'vovna Levit
, 
10.1016/j.mencom.2013.12.011
Published 2013-12-12
Communication , Volume 24, Issue 1, 35-36
16
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Vigorov A. Y. et al. Novel synthetic routes to N-(2-amino-9H-purin-6-yl)-substituted amino acids // Mendeleev Communications. 2013. Vol. 24. No. 1. pp. 35-36.
GOST all authors (up to 50) Copy
Vigorov A. Y., Krasnov V. P., Gruzdev D. A., Men'shikova A. A., Demin A. M., Levit G. L., Charushin V. N. Novel synthetic routes to N-(2-amino-9H-purin-6-yl)-substituted amino acids // Mendeleev Communications. 2013. Vol. 24. No. 1. pp. 35-36.
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TY - JOUR
DO - 10.1016/j.mencom.2013.12.011
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2013.12.011
TI - Novel synthetic routes to N-(2-amino-9H-purin-6-yl)-substituted amino acids
T2 - Mendeleev Communications
AU - Vigorov, Alexey Yur'evich
AU - Krasnov, Victor Pavlovich
AU - Gruzdev, Dmitry Andreevich
AU - Men'shikova, Alisa A
AU - Demin, Alexander Mikhailovich
AU - Levit, Galina L'vovna
AU - Charushin, Valery Nikolaevich
PY - 2013
DA - 2013/12/12
PB - Mendeleev Communications
SP - 35-36
IS - 1
VL - 24
ER -
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@article{2013_Vigorov,
author = {Alexey Yur'evich Vigorov and Victor Pavlovich Krasnov and Dmitry Andreevich Gruzdev and Alisa A Men'shikova and Alexander Mikhailovich Demin and Galina L'vovna Levit and Valery Nikolaevich Charushin},
title = {Novel synthetic routes to N-(2-amino-9H-purin-6-yl)-substituted amino acids},
journal = {Mendeleev Communications},
year = {2013},
volume = {24},
publisher = {Mendeleev Communications},
month = {Dec},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2013.12.011},
number = {1},
pages = {35--36},
doi = {10.1016/j.mencom.2013.12.011}
}
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Vigorov, Alexey Yur'evich, et al. “Novel synthetic routes to N-(2-amino-9H-purin-6-yl)-substituted amino acids.” Mendeleev Communications, vol. 24, no. 1, Dec. 2013, pp. 35-36. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2013.12.011.

Abstract

Reaction of N2-protected 2-amino-6-chloropurine with tert-butyl (S)-phenylalaninate, (R)- and (S)-valinates followed by deprotection affords 2-aminopurines bearing at 6-position the corresponding amino acid moieties, whose chiral centre is partially racemized.

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