Home / Publications / Simple and efficient synthesis of substituted 1H-indazoles

Simple and efficient synthesis of substituted 1H-indazoles

Galina Pavlovna Sagitullina 1
Galina Pavlovna Sagitullina
, 
Anna Konstantinovna Garkushenko 1
Anna Konstantinovna Garkushenko
, 
Nicolay Vladimirovich Poendaev 1
Nicolay Vladimirovich Poendaev
, 
Reva Safarovich Sagitullin 1
Reva Safarovich Sagitullin
10.1016/j.mencom.2012.05.020
Published 2012-04-27
Communication , Volume 22, Issue 3, 167-168
4
Share
Cite this
GOST
 | 
Cite this
GOST Copy
Sagitullina G. P. et al. Simple and efficient synthesis of substituted 1H-indazoles // Mendeleev Communications. 2012. Vol. 22. No. 3. pp. 167-168.
GOST all authors (up to 50) Copy
Sagitullina G. P., Garkushenko A. K., Poendaev N. V., Sagitullin R. S. Simple and efficient synthesis of substituted 1H-indazoles // Mendeleev Communications. 2012. Vol. 22. No. 3. pp. 167-168.
RIS
 | 
Cite this
RIS Copy
TY - JOUR
DO - 10.1016/j.mencom.2012.05.020
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2012.05.020
TI - Simple and efficient synthesis of substituted 1H-indazoles
T2 - Mendeleev Communications
AU - Sagitullina, Galina Pavlovna
AU - Garkushenko, Anna Konstantinovna
AU - Poendaev, Nicolay Vladimirovich
AU - Sagitullin, Reva Safarovich
PY - 2012
DA - 2012/04/27
PB - Mendeleev Communications
SP - 167-168
IS - 3
VL - 22
ER -
BibTex
 | 
Cite this
BibTex (up to 50 authors) Copy
@article{2012_Sagitullina,
author = {Galina Pavlovna Sagitullina and Anna Konstantinovna Garkushenko and Nicolay Vladimirovich Poendaev and Reva Safarovich Sagitullin},
title = {Simple and efficient synthesis of substituted 1H-indazoles},
journal = {Mendeleev Communications},
year = {2012},
volume = {22},
publisher = {Mendeleev Communications},
month = {Apr},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2012.05.020},
number = {3},
pages = {167--168},
doi = {10.1016/j.mencom.2012.05.020}
}
MLA
Cite this
MLA Copy
Sagitullina, Galina Pavlovna, et al. “Simple and efficient synthesis of substituted 1H-indazoles.” Mendeleev Communications, vol. 22, no. 3, Apr. 2012, pp. 167-168. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2012.05.020.

Abstract

3-Aryl-5-aroylindazoles were prepared by a simple two-stage protocol from 3,5-diaroyl-2,6-dimethylpyridines.

References

1.
10.1016/j.mencom.2012.05.020_bib0005
Wermuth
Compr. Med. Chem. II, 2006
3.
Isolation and structure determination of nigellicine, a novel alkaloid from the seeds of
Atta-ur-Rahman, Malik S., Cun-heng H., Clardy J.
Tetrahedron Letters, 1985
4.
Nigellidine — A new indazole alkaloid from the seeds of Nigella sativa
Atta-ur-Rahman, Malik S., Hasan S.S., Choudhary M.I., Ni C., Clardy J.
Tetrahedron Letters, 1995
7.
Bendazac Lysine
Balfour J.A., Clissold S.P.
Drugs, 1990
8.
Radical scavenger activity of bendazac, an anticataract non-steroidal anti-inflammatory agent
Guglielmotti A., Capezzone de Joannon A., Cazzolla N., Marchetti M., Soldo L., Cavallo G., Pinza M.
Pharmacological Research, 1995
10.
Photoallergic contact dermatitis from benzydamine presenting mainly as lip dermatitis
Canelas M.M., Cardoso J.C., Gonçalo M., Figueiredo A.
Contact Dermatitis, 2010
11.
Glycolysis inhibition for anticancer treatment
Pelicano H., Martin D.S., Xu R., Huang P.
Oncogene, 2006
12.
The anti-inflammatory agent bindarit inhibits neointima formation in both rats and hyperlipidaemic mice
Grassia G., Maddaluno M., Guglielmotti A., Mangano G., Biondi G., Maffia P., Ialenti A.
Cardiovascular Research, 2009
13.
Treatment with bindarit, a blocker of MCP-1 synthesis, protects mice against acute pancreatitis
Bhatia M., Ramnath R.D., Chevali L., Guglielmotti A.
American Journal of Physiology - Gastrointestinal and Liver Physiology, 2005
14.
Granisetron
Plosker G.L., Goa K.L.
Drugs, 1991
16.
xxx, http://www.genengnews.com.
17.
Recent Advances in the Chemistry of Indazoles
Schmidt A., Beutler A., Snovydovych B.
European Journal of Organic Chemistry, 2008
18.
W. Stadlbauer, Science of Synthesis: Houben-Weyl Methods of Molecular Transformations, Georg Thieme Verlag, Stuttgart, New York, 2007, vol. 12, p. 227.
19.
10.1016/j.mencom.2012.05.020_bib0095
Cottyn
Synlett, 2007
20.
Synthesis of 3-Substituted Indazoles from Arynes and N-Tosylhydrazones
Li P., Zhao J., Wu C., Larock R.C., Shi F.
Organic Letters, 2011
21.
One-pot synthesis of 1-alkyl-1H-indazoles from 1,1-dialkylhydrazones via aryne annulation
Markina N.A., Dubrovskiy A.V., Larock R.C.
Organic and Biomolecular Chemistry, 2012
22.
Synthesis of New 1H-Indazoles through Diels-Alder Transformations of 4-Styrylpyrazoles under Microwave Irradiation Conditions
Silva V.L., Silva A.M., Pinto D.C., Elguero J., Cavaleiro J.A.
European Journal of Organic Chemistry, 2009
23.
Efficient Synthesis of 3-Substituted Indazoles Using Pd-Catalyzed Intramolecular Amination Reaction ofN-Tosylhydrazones
Inamoto K., Katsuno M., Yoshino T., Suzuki I., Hiroya K., Sakamoto T.
Chemistry Letters, 2004
24.
The synthesis of substituted indazolesviacyclization of various hydrazones in the presence of polyphosphoric acid (PPA)
Guofu Q., Jiangtao S., Xichun F., Lamei W., Wenjin X., Xianming H.
Journal of Heterocyclic Chemistry, 2004
25.
Reactions of hydroxybenzophenone with hydrazines
Krishnan R., Lang S.A., Lin Y., Wilkinson R.G.
Journal of Heterocyclic Chemistry, 1988
27.
A. K. Garkushenko, N.V. Poendaev, M.A. Vorontsova and G. P. Sagitullina, Khim. Geterotsikl. Soedin., 2011, 573.[Chem. Heterocycl. Compd. (Engl. Transl.), 2011, 47, 470].
28.
A. K. Garkushenko, M.A. Makarova, O.P. Sorokina, N.V. Poendaev, M.A. Vorontsova and G. P. Sagitullina, Khim. Geterotsikl. Soedin., 2011, 586.[Chem. Heterocycl. Compd. (Engl. Transl.), 2011, 47, 482].
29.
Recyclization of polysubstituted pyridinium salts
Shkil G.P., Lusis V., Muceniece D., Sagitullin R.S.
Tetrahedron, 1995