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Synthesis of diglyceride conjugate of selectin ligand SiaLeX as a vector for targeting of drug-loaded liposomes

Elena L'vovna Vodovozova 1
Elena L'vovna Vodovozova
, 
Galina Valentinovna Pazynina 1
Galina Valentinovna Pazynina
, 
10.1016/j.mencom.2011.03.002
Published 2011-03-10
Communication , Volume 21, Issue 2, 69-71
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Vodovozova E. L., Pazynina G. V., Bovin N. V. Synthesis of diglyceride conjugate of selectin ligand SiaLeX as a vector for targeting of drug-loaded liposomes // Mendeleev Communications. 2011. Vol. 21. No. 2. pp. 69-71.
GOST all authors (up to 50) Copy
Vodovozova E. L., Pazynina G. V., Bovin N. V. Synthesis of diglyceride conjugate of selectin ligand SiaLeX as a vector for targeting of drug-loaded liposomes // Mendeleev Communications. 2011. Vol. 21. No. 2. pp. 69-71.
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TY - JOUR
DO - 10.1016/j.mencom.2011.03.002
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2011.03.002
TI - Synthesis of diglyceride conjugate of selectin ligand SiaLeX as a vector for targeting of drug-loaded liposomes
T2 - Mendeleev Communications
AU - Vodovozova, Elena L'vovna
AU - Pazynina, Galina Valentinovna
AU - Bovin, Nicolai Vladimirovich
PY - 2011
DA - 2011/03/10
PB - Mendeleev Communications
SP - 69-71
IS - 2
VL - 21
ER -
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@article{2011_Vodovozova,
author = {Elena L'vovna Vodovozova and Galina Valentinovna Pazynina and Nicolai Vladimirovich Bovin},
title = {Synthesis of diglyceride conjugate of selectin ligand SiaLeX as a vector for targeting of drug-loaded liposomes},
journal = {Mendeleev Communications},
year = {2011},
volume = {21},
publisher = {Mendeleev Communications},
month = {Mar},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2011.03.002},
number = {2},
pages = {69--71},
doi = {10.1016/j.mencom.2011.03.002}
}
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Vodovozova, Elena L'vovna, et al. “Synthesis of diglyceride conjugate of selectin ligand SiaLeX as a vector for targeting of drug-loaded liposomes.” Mendeleev Communications, vol. 21, no. 2, Mar. 2011, pp. 69-71. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2011.03.002.

Abstract

A conjugate of tetrasaccharide Sialyl Lewis X [SiaLeX, Neu5Acα2-3Galβ1-4(Fucα1-3)GlcNAcβ] 3-aminopropyl glycoside and rac-1,2-dioleoyl-3-carboxymethylene[poly(8–15)oxyethylene]oxyacetylamidopropionylglycerol amenable for the incorporation in lipid bilayer of drug-loaded liposomes to achieve targeting in tumors and inflammation foci was obtained by the formation of carboxamide bond.

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