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Synthesis of 5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo-[3,2-b]pyridine-3-carboxylic acids by three-component condensation of 3-aminopyrrole derivatives

Boris Valer'evich Lichitsky 1
Boris Valer'evich Lichitsky
, 
Arkady Anatol'evich Dudinov 1
Arkady Anatol'evich Dudinov
, 
Andrey Nikolaevich Komogortsev 1
Andrey Nikolaevich Komogortsev
, 
Mikhail Mikhailovich Krayushkin 1
Mikhail Mikhailovich Krayushkin
10.1016/j.mencom.2010.09.004
Published 2010-09-09
Communication , Volume 20, Issue 5, 255-256
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Lichitsky B. V. et al. Synthesis of 5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo-[3,2-b]pyridine-3-carboxylic acids by three-component condensation of 3-aminopyrrole derivatives // Mendeleev Communications. 2010. Vol. 20. No. 5. pp. 255-256.
GOST all authors (up to 50) Copy
Lichitsky B. V., Dudinov A. A., Komogortsev A. N., Krayushkin M. M. Synthesis of 5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo-[3,2-b]pyridine-3-carboxylic acids by three-component condensation of 3-aminopyrrole derivatives // Mendeleev Communications. 2010. Vol. 20. No. 5. pp. 255-256.
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TY - JOUR
DO - 10.1016/j.mencom.2010.09.004
UR - https://mendcomm.colab.ws/publications/10.1016/j.mencom.2010.09.004
TI - Synthesis of 5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo-[3,2-b]pyridine-3-carboxylic acids by three-component condensation of 3-aminopyrrole derivatives
T2 - Mendeleev Communications
AU - Lichitsky, Boris Valer'evich
AU - Dudinov, Arkady Anatol'evich
AU - Komogortsev, Andrey Nikolaevich
AU - Krayushkin, Mikhail Mikhailovich
PY - 2010
DA - 2010/09/09
PB - Mendeleev Communications
SP - 255-256
IS - 5
VL - 20
ER -
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@article{2010_Lichitsky,
author = {Boris Valer'evich Lichitsky and Arkady Anatol'evich Dudinov and Andrey Nikolaevich Komogortsev and Mikhail Mikhailovich Krayushkin},
title = {Synthesis of 5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo-[3,2-b]pyridine-3-carboxylic acids by three-component condensation of 3-aminopyrrole derivatives},
journal = {Mendeleev Communications},
year = {2010},
volume = {20},
publisher = {Mendeleev Communications},
month = {Sep},
url = {https://mendcomm.colab.ws/publications/10.1016/j.mencom.2010.09.004},
number = {5},
pages = {255--256},
doi = {10.1016/j.mencom.2010.09.004}
}
MLA
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Lichitsky, Boris Valer'evich, et al. “Synthesis of 5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo-[3,2-b]pyridine-3-carboxylic acids by three-component condensation of 3-aminopyrrole derivatives.” Mendeleev Communications, vol. 20, no. 5, Sep. 2010, pp. 255-256. https://mendcomm.colab.ws/publications/10.1016/j.mencom.2010.09.004.

Abstract

5-Oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-b]pyridine-3-carboxylic acids were prepared by three-component condensation of 3-aminopyrroles, (het)aromatic aldehydes and Meldrum's acid. The labile intermediate 3-aminopyrrole derivative was generated in situ by regioselective (at 2-position) decarboxylation of 3-aminopyrrole-2,4-dicarboxylic acid.

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